Assay Detail
Binding
CHEMBL5147294
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of tyrosinase (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Polyphenolic compounds: Synthesis, assessment of antimicrobial effect and enzymes inhibition against important medicinal enzymes with computational details.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.22 | 4.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL50 | QUERCETIN | 3.0 | 1 | 4.35 |
| CHEMBL150 | KAEMPFEROL | 1.0 | 1 | 4.19 |
| CHEMBL266564 | TILIROSIDE | — | 1 | 4.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL50 | QUERCETIN | IC50 | = | 44380.0 | nM | 4.35 |
| CHEMBL150 | KAEMPFEROL | IC50 | = | 65110.0 | nM | 4.19 |
| CHEMBL266564 | TILIROSIDE | IC50 | = | 78530.0 | nM | 4.11 |