Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5147983

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HIV-1 JRFL assessed as inhibition of viral growth
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human immunodeficiency virus 1
Confidence 1 — Organism
Curated By Autocuration

Target

Human immunodeficiency virus 1 (CHEMBL378)
Type ORGANISM
Organism Human immunodeficiency virus 1

Publication

Development of Azaindole-Based Frameworks as Potential Antiviral Agents and Their Future Perspectives.
Urvashi, Senthil Kumar JB, Das P, Tandon V.
J Med Chem (2022) 65 : 6454 -6495
PubMed 35477274 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 9.84 10.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL236995 1 10.30
CHEMBL2332337 1 10.15
CHEMBL238103 1 9.06

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL236995 EC50 = 0.05 nM 10.30
CHEMBL2332337 EC50 = 0.07 nM 10.15
CHEMBL238103 EC50 = 0.88 nM 9.06