Assay Detail
Binding
CHEMBL5149210
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [18F]-LU13 from human CB2 receptor transfected in CHO cells membrane homogenate incubated for 90 mins by competitive radioligand binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Subcellular | Membrane |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structure-Based Design, Optimization, and Development of [<sup>18</sup>F]LU13: A Novel Radioligand for Cannabinoid Receptor Type 2 Imaging in the Brain with PET.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.93 | 8.93 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5198892 | — | — | 1 | 8.93 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5198892 | — | IC50 | = | 1.17 | nM | 8.93 |