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Assay Detail

CHEMBL5155632

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against mouse RAW264.7 cells measured after 72 hrs by SRB assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Identification and optimization of biphenyl derivatives as novel tubulin inhibitors targeting colchicine-binding site overcoming multidrug resistance.
Cheng B, Zhu G, Meng L, Wu G, Chen Q, Ma S.
Eur J Med Chem (2022) 228 : 113930 -113930
PubMed 34794817 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 8.12 8.12

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5206531 1 8.12

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5206531 IC50 = 7.6 nM 8.12