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Assay Detail

CHEMBL5157985

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Agonist activity at S1P1 receptor (unknown origin) expressed in PathHunter HEK 293 EDG1 Total GPCR Internalization cells assessed as receptor internalization incubated for 90 mins by measuring chemiluminescence signal by microplate reader method
65
Total Activities
65
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type PathHunter HEK 293 EDG1 Total GPCR Internalization
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sphingosine 1-phosphate receptor 1 (CHEMBL4333)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of Novel Sphingosine-1-Phosphate-1 Receptor Agonists for the Treatment of Multiple Sclerosis.
Park SJ, Yeon SK, Kim Y, Kim HJ, Kim S, Kim J, Choi JW, Kim B, Lee EH, Kim R, Seo SH, Lee J, Kim JW, Lee HY, Hwang H, Bahn YS, Cheong E, Park JH, Park KD.
J Med Chem (2022) 65 : 3539 -3562
PubMed 35077170 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 65 7.26 9.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL114606 1 9.15
CHEMBL5170826 1 9.08
CHEMBL5172303 1 8.65
CHEMBL5177759 1 8.59
CHEMBL5174924 1 8.50
CHEMBL5179798 1 8.39
CHEMBL5183779 1 8.29
CHEMBL5176185 1 7.96
CHEMBL5176383 1 7.93
CHEMBL5202775 1 7.86
CHEMBL5198753 1 7.84
CHEMBL5173103 1 7.78
CHEMBL5178933 1 7.61
CHEMBL5204567 1 7.60
CHEMBL5196884 1 7.52
CHEMBL5173606 1 7.46
CHEMBL5182813 1 7.44
CHEMBL5186672 1 7.42
CHEMBL5197074 1 7.34
CHEMBL5177232 1 7.20
CHEMBL5202986 1 7.18
CHEMBL5192922 1 7.09
CHEMBL5189040 1 6.97
CHEMBL5182920 1 6.96
CHEMBL5178428 1 6.96
CHEMBL5201690 1 6.95
CHEMBL5199664 1 6.91
CHEMBL5202350 1 6.84
CHEMBL5192549 1 6.82
CHEMBL5169412 1 6.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL114606 EC50 = 0.7 nM 9.15
CHEMBL5170826 EC50 = 0.84 nM 9.08
CHEMBL5172303 EC50 = 2.25 nM 8.65
CHEMBL5177759 EC50 = 2.59 nM 8.59
CHEMBL5174924 EC50 = 3.16 nM 8.50
CHEMBL5179798 EC50 = 4.06 nM 8.39
CHEMBL5183779 EC50 = 5.09 nM 8.29
CHEMBL5176185 EC50 = 11.1 nM 7.96
CHEMBL5176383 EC50 = 11.8 nM 7.93
CHEMBL5202775 EC50 = 13.8 nM 7.86
CHEMBL5198753 EC50 = 14.3 nM 7.84
CHEMBL5173103 EC50 = 16.8 nM 7.78
CHEMBL5178933 EC50 = 24.6 nM 7.61
CHEMBL5204567 EC50 = 25.0 nM 7.60
CHEMBL5196884 EC50 = 30.5 nM 7.52
CHEMBL5173606 EC50 = 34.6 nM 7.46
CHEMBL5182813 EC50 = 36.4 nM 7.44
CHEMBL5186672 EC50 = 38.5 nM 7.42
CHEMBL5197074 EC50 = 45.3 nM 7.34
CHEMBL5177232 EC50 = 63.2 nM 7.20
CHEMBL5202986 EC50 = 66.5 nM 7.18
CHEMBL5192922 EC50 = 80.6 nM 7.09
CHEMBL5189040 EC50 = 106.0 nM 6.97
CHEMBL5182920 EC50 = 111.0 nM 6.96
CHEMBL5178428 EC50 = 111.0 nM 6.96
CHEMBL5201690 EC50 = 112.0 nM 6.95
CHEMBL5199664 EC50 = 122.0 nM 6.91
CHEMBL5202350 EC50 = 146.0 nM 6.84
CHEMBL5192549 EC50 = 152.0 nM 6.82
CHEMBL5169412 EC50 = 160.0 nM 6.80
CHEMBL5183758 EC50 = 209.0 nM 6.68
CHEMBL5203930 EC50 = 237.0 nM 6.62
CHEMBL5201117 EC50 = 283.0 nM 6.55
CHEMBL5176091 EC50 = 286.0 nM 6.54
CHEMBL5186304 EC50 = 313.0 nM 6.50
CHEMBL5191622 EC50 = 346.0 nM 6.46
CHEMBL5194896 EC50 = 378.0 nM 6.42
CHEMBL5185995 EC50 = 385.0 nM 6.42
CHEMBL5187844 EC50 = 414.0 nM 6.38
CHEMBL5203643 EC50 = 594.0 nM 6.23
CHEMBL5172318 EC50 = 813.0 nM 6.09
CHEMBL5181453 EC50 = 876.0 nM 6.06
CHEMBL5208384 EC50 = 973.0 nM 6.01
CHEMBL5180613 EC50 > 1000.0 nM -
CHEMBL5180579 EC50 > 1000.0 nM -
CHEMBL5180309 EC50 > 1000.0 nM -
CHEMBL5173741 EC50 > 1000.0 nM -
CHEMBL5186460 EC50 > 1000.0 nM -
CHEMBL5191394 EC50 > 1000.0 nM -
CHEMBL5209429 EC50 > 1000.0 nM -