Assay Detail

CHEMBL5213823

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Binding

Selectivity interaction (GPCR panel (PDSP screen)) EUB0000735a ADRB1

ChEMBL ↗

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Target

Beta-1 adrenergic receptor (CHEMBL213) ↗

Open DB target context

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Beta-1 adrenergic receptor (CHEMBL213) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Beta-1 adrenergic receptor

CHEMBL213

Anchored from Assay target.

Protein identity Beta-1 adrenergic receptor

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Homo sapiens
Category	Selectivity assay
Confidence	9 — Direct single protein target
Curated By	Autocuration

Target

Beta-1 adrenergic receptor (CHEMBL213) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Selectivity Literature for EUbOPEN Chemogenomics Library wave 3

EUbOPEN
(2023)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
Ki	1	5.26	5.26

Assay Parameters

Parameter	Type	Value	Units	Text
Protein family	Protein family	-	—	GPCR

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL3617968	BAY-678	—	1	5.26

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL3617968	BAY-678	Ki	=	5450.0	nM	5.26