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Assay Detail

CHEMBL5214074

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Selectivity interaction (HAT panel) EUB0000329a MYST3
1
Total Activities
1
Compounds Tested
1
Activity Types
1
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Category Selectivity assay
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Histone acetyltransferase KAT6A (CHEMBL3774298)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Selectivity Literature for EUbOPEN Chemogenomics Library wave 3
EUbOPEN
(2023)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.43 7.43

Assay Parameters

Parameter Type Value Units Text
Protein family Protein family - HAT

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4456585 WM-1119 1 7.43

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4456585 WM-1119 IC50 = 37.0 nM 7.43