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Assay Detail

CHEMBL5217153

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of His-tagged human LMW-PTP expressed in Escherichia coli BL21 using pNPP as substrate incubated for 10 mins by microplate reader based spectrophotometric analysis
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Publication

Structure-Based Design of Active-Site-Directed, Highly Potent, Selective, and Orally Bioavailable Low-Molecular-Weight Protein Tyrosine Phosphatase Inhibitors.
He R, Wang J, Yu ZH, Moyers JS, Michael MD, Durham TB, Cramer JW, Qian Y, Lin A, Wu L, Noinaj N, Barrett DG, Zhang ZY.
J Med Chem (2022) 65 : 13892 -13909
PubMed 36197449 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 30 6.00 8.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5218807 1 8.40
CHEMBL5219822 1 8.10
CHEMBL5218783 1 7.31
CHEMBL5220687 1 7.25
CHEMBL5220615 1 6.92
CHEMBL5220051 1 6.70
CHEMBL5218478 1 6.52
CHEMBL5219403 1 6.52
CHEMBL5219065 1 6.40
CHEMBL5218609 1 6.40
CHEMBL5218798 1 6.22
CHEMBL5218883 1 5.92
CHEMBL5221084 1 5.82
CHEMBL5220114 1 5.82
CHEMBL5219085 1 5.82
CHEMBL5219469 1 5.82
CHEMBL5219423 1 5.77
CHEMBL5219519 1 5.66
CHEMBL5220487 1 5.47
CHEMBL5219635 1 5.47
CHEMBL5220131 1 5.36
CHEMBL5219411 1 5.28
CHEMBL5219998 1 5.27
CHEMBL5219580 1 5.22
CHEMBL5220369 1 5.22
CHEMBL5220894 1 5.07
CHEMBL5218748 1 4.94
CHEMBL5219215 1 4.91
CHEMBL5219416 1 4.52
CHEMBL5218939 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5218807 IC50 = 4.0 nM 8.40
CHEMBL5219822 IC50 = 8.0 nM 8.10
CHEMBL5218783 IC50 = 49.0 nM 7.31
CHEMBL5220687 IC50 = 56.0 nM 7.25
CHEMBL5220615 IC50 = 121.0 nM 6.92
CHEMBL5220051 IC50 = 200.0 nM 6.70
CHEMBL5218478 IC50 = 300.0 nM 6.52
CHEMBL5219403 IC50 = 300.0 nM 6.52
CHEMBL5219065 IC50 = 400.0 nM 6.40
CHEMBL5218609 IC50 = 400.0 nM 6.40
CHEMBL5218798 IC50 = 600.0 nM 6.22
CHEMBL5218883 IC50 = 1200.0 nM 5.92
CHEMBL5221084 IC50 = 1500.0 nM 5.82
CHEMBL5220114 IC50 = 1500.0 nM 5.82
CHEMBL5219085 IC50 = 1500.0 nM 5.82
CHEMBL5219469 IC50 = 1500.0 nM 5.82
CHEMBL5219423 IC50 = 1700.0 nM 5.77
CHEMBL5219519 IC50 = 2200.0 nM 5.66
CHEMBL5220487 IC50 = 3400.0 nM 5.47
CHEMBL5219635 IC50 = 3400.0 nM 5.47
CHEMBL5220131 IC50 = 4400.0 nM 5.36
CHEMBL5219411 IC50 = 5200.0 nM 5.28
CHEMBL5219998 IC50 = 5400.0 nM 5.27
CHEMBL5219580 IC50 = 6000.0 nM 5.22
CHEMBL5220369 IC50 = 6000.0 nM 5.22
CHEMBL5220894 IC50 = 8600.0 nM 5.07
CHEMBL5218748 IC50 = 11400.0 nM 4.94
CHEMBL5219215 IC50 = 12200.0 nM 4.91
CHEMBL5219416 IC50 = 30000.0 nM 4.52
CHEMBL5218939 IC50 > 100000.0 nM -