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Assay Detail

CHEMBL5217447

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of bovine GGT1 transpeptidation using gamma-glutamyl-p-nitroanilide in presence of Gly-Gly
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Bos taurus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Design and evaluation of novel analogs of 2-amino-4-boronobutanoic acid (ABBA) as inhibitors of human gamma-glutamyl transpeptidase.
Nguyen L, Schultz DC, Terzyan SS, Rezaei M, Songb J, Li C, You Y, Hanigan MH.
Bioorg Med Chem (2022) 73 : 116986 -116986
PubMed 36208545 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.77 7.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5220943 1 7.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5220943 Ki = 17.0 nM 7.77