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Assay Detail

CHEMBL5223280

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of recombinant West Nile virus NS2B-NS3 protease using Pyr-RTKR-AMC as substrate assessed as change in fluorescence intensity preincubated for 15 mins followed by substrate addition by fluorescence based microplate reader analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism West Nile virus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Genome polyprotein (CHEMBL5419)
Type SINGLE PROTEIN
Organism West Nile virus

Publication

Targeting the protease of West Nile virus.
Voss S, Nitsche C.
RSC Med Chem (2021) 12 : 1262 -1272
PubMed 34458734 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.21 5.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3344319 1 5.21

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3344319 IC50 = 6100.0 nM 5.21