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Assay Detail

CHEMBL5226964

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of NO production in LPS-stimulated mouse RAW264.7 cells preincubated with compound for 30 mins followed by LPS stimulation and measured after 24 hrs by Griess reagent-based assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Discovery of natural anti-inflammatory alkaloids: Potential leads for the drug discovery for the treatment of inflammation.
Bai R, Yao C, Zhong Z, Ge J, Bai Z, Ye X, Xie T, Xie Y.
Eur J Med Chem (2021) 213 : 113165 -113165
PubMed 33454546 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.75 5.17

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2018557 1 5.17
CHEMBL458702 DECARINE 1 4.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2018557 IC50 = 6800.0 nM 5.17
CHEMBL458702 DECARINE IC50 = 48400.0 nM 4.32