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Assay Detail

CHEMBL5230042

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Cytotoxicity against LPS-stimulated mouse RAW264.7 cells assessed as cell growth inhibition preincubated for 15 mins followed by LPS stimulation and measured after 20 hrs by CCK-8 assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Anti-inflammatory Quinoline Alkaloids from the Roots of <i>Waltheria indica</i>.
Liu F, O'Donnell TJ, Park EJ, Kovacs S, Nakamura K, Dave A, Luo Y, Sun R, Wall M, Wongwiwatthananukit S, Silva DK, Williams PG, Pezzuto JM, Chang LC.
J Nat Prod (2023) 86 : 276 -289
PubMed 36746775 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.52 4.59

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5267196 1 4.59
CHEMBL3342751 1 4.49
CHEMBL5291228 1 4.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5267196 IC50 = 25900.0 nM 4.59
CHEMBL3342751 IC50 = 32200.0 nM 4.49
CHEMBL5291228 IC50 = 33300.0 nM 4.48