Assay Detail
Binding
CHEMBL5231297
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of SMARCA2 BD (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Probable global transcription activator SNF2L2 (CHEMBL2362979) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.27 | 6.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4746865 | — | — | 1 | 6.43 |
| CHEMBL5278697 | — | — | 1 | 6.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4746865 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL5278697 | — | IC50 | = | 770.0 | nM | 6.11 |