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Assay Detail

CHEMBL5232209

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Cytotoxicity against mouse NIH/3T3 cells assessed as reduction in cell viability incubated for 4 days by SRB assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Mus musculus
Cell Type NIH3T3
Confidence 1 — Organism
Curated By Autocuration

Target

NIH3T3 (CHEMBL614822)
Type CELL-LINE
Organism Mus musculus

Publication

Inhibitors of Eukaryotic Translational Machinery as Therapeutic Agents.
Fan A, Sharp PP.
J Med Chem (2021) 64 : 2436 -2465
PubMed 33592144 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 8.38 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5268659 1 8.70
CHEMBL2058177 1 8.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5268659 IC50 = 2.0 nM 8.70
CHEMBL2058177 IC50 = 9.0 nM 8.05