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Assay Detail

CHEMBL5232732

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to human Arg II
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Arginase-2, mitochondrial (CHEMBL1795148)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Targeting Metalloenzymes by Boron-Containing Metal-Binding Pharmacophores.
Xiao YC, Yu JL, Dai QQ, Li G, Li GB.
J Med Chem (2021) 64 : 17706 -17727
PubMed 34875836 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.05 7.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL539140 1 7.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL539140 Ki = 89.0 nM 7.05