Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5235226

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Cytotoxicity against mouse RAW264.7 cells assessed as reduction in cell viability by MTT assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Anti-inflammatory activity of naturally occuring diarylheptanoids - A review.
Vanucci-Bacqué C, Bedos-Belval F.
Bioorg Med Chem (2021) 31 : 115971 -115971
PubMed 33422907 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.60 5.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5276513 1 5.05
CHEMBL330645 PLATYPHYLLENONE 1 4.51
CHEMBL2346808 1 4.44
CHEMBL464274 DEHYDROHIRSUTANONOL 1 4.41

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5276513 IC50 = 9000.0 nM 5.05
CHEMBL330645 PLATYPHYLLENONE IC50 = 30700.0 nM 4.51
CHEMBL2346808 IC50 = 36400.0 nM 4.44
CHEMBL464274 DEHYDROHIRSUTANONOL IC50 = 39000.0 nM 4.41