Assay Detail
Functional
CHEMBL5236763
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Antiproliferative activity against human HCT-116 cells assessed as inhibition of cell proliferation incubated for 24 hrs by MTT assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HCT-116 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Furazans in Medicinal Chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 4.88 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5187860 | — | — | 1 | 5.80 |
| CHEMBL3589160 | — | — | 1 | 4.51 |
| CHEMBL4451478 | — | — | 1 | 4.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5187860 | — | EC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL3589160 | — | EC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL4451478 | — | EC50 | = | 45800.0 | nM | 4.34 |