Assay Detail
Binding
CHEMBL5237491
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PAR2 expressed in human HT-29 cells incubated for 30 mins by FLIPR Tetra system method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HT-29 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Imidazo[1,2-b]pyridazine as privileged scaffold in medicinal chemistry: An extensive review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 9.15 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5273903 | — | — | 1 | 9.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5273903 | — | IC50 | = | 0.7 | nM | 9.15 |