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Assay Detail

CHEMBL5237882

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HIV-1 infected in human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assay
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human immunodeficiency virus 1
Cell Type C8166
Confidence 1 — Organism
Curated By Autocuration

Target

Human immunodeficiency virus 1 (CHEMBL378)
Type ORGANISM
Organism Human immunodeficiency virus 1

Publication

Bioactive Aurones, Indanones, and Other Hemiindigoid Scaffolds: Medicinal Chemistry and Photopharmacology Perspectives.
Lazinski LM, Royal G, Robin M, Maresca M, Haudecoeur R.
J Med Chem (2022) 65 : 12594 -12625
PubMed 36126323 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.62 5.62
EC50 1 4.92 4.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5267841 1 5.62
CHEMBL3298066 1 4.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5267841 IC50 = 2400.0 nM 5.62
CHEMBL3298066 EC50 = 12000.0 nM 4.92