Assay Detail
Binding
CHEMBL5239289
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to GST tagged AR LBD (unknown orign) by radioligand binding assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
A Comprehensive Overview of Small-Molecule Androgen Receptor Degraders: Recent Progress and Future Perspectives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.84 | 7.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4584527 | — | — | 1 | 7.11 |
| CHEMBL4444904 | — | — | 1 | 6.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4584527 | — | Ki | = | 78.06 | nM | 7.11 |
| CHEMBL4444904 | — | Ki | = | 267.39 | nM | 6.57 |