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Assay Detail

CHEMBL5247261

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Influenza A virus A/PR/8/34 (PR8) strain infected in MDCK cells assessed as reduction in viral infection incubated for 72 hrs by crystal violet staining based assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Influenza A virus
Confidence 1 — Organism
Curated By Autocuration

Target

Influenza A virus (CHEMBL613740)
Type ORGANISM
Organism Influenza A virus

Publication

Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design.
Subbaiah MAM, Meanwell NA.
J Med Chem (2021) 64 : 14046 -14128
PubMed 34591488 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.41 6.48

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2040554 1 6.48
CHEMBL5286364 1 5.96
CHEMBL467389 1 4.67
CHEMBL2040641 1 4.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2040554 IC50 = 330.0 nM 6.48
CHEMBL5286364 IC50 = 1100.0 nM 5.96
CHEMBL467389 IC50 = 21300.0 nM 4.67
CHEMBL2040641 IC50 = 29400.0 nM 4.53