Assay Detail
Binding
CHEMBL5259644
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Agonist activity at GPR-35 (unknown origin) expressed in HT-29 cells by DMR assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HT-29 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development and Characterization of Fluorescent Probes for the G Protein-Coupled Receptor 35.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 7.40 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL177880 | PAMOIC ACID | — | 1 | 8.52 |
| CHEMBL428880 | CROMOLYN | 4.0 | 1 | 6.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL177880 | PAMOIC ACID | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL428880 | CROMOLYN | EC50 | = | 520.0 | nM | 6.28 |