Assay Detail
Functional
CHEMBL5261663
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Cytotoxicity against human EOL1 cells measured after 8 days
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | EOL1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Inhibition of bromodomain-containing protein 9 for the prevention of epigenetically-defined drug resistance.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.79 | 6.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5270178 | — | — | 1 | 6.02 |
| CHEMBL5268484 | — | — | 1 | 5.87 |
| CHEMBL5282240 | — | — | 1 | 5.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5270178 | — | IC50 | = | 950.0 | nM | 6.02 |
| CHEMBL5268484 | — | IC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL5282240 | — | IC50 | = | 3300.0 | nM | 5.48 |