Assay Detail
Binding
CHEMBL5265013
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at PPARdelta (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Peroxisome proliferator-activated receptor delta (CHEMBL3979) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Emerging targets and potential therapeutic agents in non-alcoholic fatty liver disease treatment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 8.00 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL230158 | SELADELPAR | 4.0 | 1 | 8.70 |
| CHEMBL153057 | — | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL230158 | SELADELPAR | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL153057 | — | EC50 | = | 50.0 | nM | 7.30 |