Assay Detail
Functional
CHEMBL5304677
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Measurement of the ATPase catalytic activity using the ADP-Glo detection (SMARCA2)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Probable global transcription activator SNF2L2 (CHEMBL2362979) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe FHT-2344
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.80 | 7.86 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5308262 | — | — | 1 | 7.86 |
| CHEMBL5306285 | — | — | 1 | 5.73 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5308262 | — | IC50 | = | 13.8 | nM | 7.86 |
| CHEMBL5306285 | — | IC50 | = | 1880.0 | nM | 5.73 |