Assay Detail
Binding
CHEMBL5316849
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Inhibition of PKD1 (unknown origin)
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Small Molecule Inhibitors of Protein Kinase D: Early Development, Current Approaches, and Future Directions.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 7.05 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5440043 | — | — | 1 | 9.00 |
| CHEMBL5419827 | — | — | 1 | 9.00 |
| CHEMBL5428541 | — | — | 1 | 9.00 |
| CHEMBL281948 | K-252A | — | 1 | 8.15 |
| CHEMBL5413306 | — | — | 1 | 7.80 |
| CHEMBL302449 | GO-6976 | — | 1 | 7.70 |
| CHEMBL388978 | STAUROSPORINE | — | 1 | 7.40 |
| CHEMBL5398617 | — | — | 1 | 7.28 |
| CHEMBL238125 | — | — | 1 | 6.97 |
| CHEMBL264406 | — | — | 1 | 6.81 |
| CHEMBL471474 | HYPOTHEMYCIN | — | 1 | 6.30 |
| CHEMBL5434569 | — | — | 1 | 5.99 |
| CHEMBL5432054 | — | — | 1 | 5.63 |
| CHEMBL5399250 | — | — | 1 | 5.62 |
| CHEMBL1504776 | — | — | 1 | 5.50 |
| CHEMBL261491 | — | — | 1 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5440043 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5419827 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5428541 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL281948 | K-252A | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL5413306 | — | IC50 | = | 16.0 | nM | 7.80 |
| CHEMBL302449 | GO-6976 | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL388978 | STAUROSPORINE | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL5398617 | — | IC50 | = | 53.0 | nM | 7.28 |
| CHEMBL238125 | — | IC50 | = | 106.0 | nM | 6.97 |
| CHEMBL264406 | — | IC50 | = | 155.0 | nM | 6.81 |
| CHEMBL471474 | HYPOTHEMYCIN | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL5434569 | — | IC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL5432054 | — | IC50 | = | 2340.0 | nM | 5.63 |
| CHEMBL5399250 | — | IC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL1504776 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL261491 | — | IC50 | = | 20000.0 | nM | 4.70 |