Assay Detail
Functional
CHEMBL5320600
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Antitumor activity against human CNE cells assessed as cell growth inhibition
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CNE |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
From Natural Sources to Synthetic Derivatives: The Allyl Motif as a Powerful Tool for Fragment-Based Design in Cancer Treatment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.75 | 4.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4436520 | — | — | 1 | 4.75 |
| CHEMBL4469205 | — | — | 1 | 4.74 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4436520 | — | IC50 | = | 17800.0 | nM | 4.75 |
| CHEMBL4469205 | — | IC50 | = | 18300.0 | nM | 4.74 |