Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5325841

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HCT-116 cells assessed as reduction in cell viability measured after 48 hrs
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HCT-116
Confidence 1 — Organism
Curated By Autocuration

Target

HCT-116 (CHEMBL394)
Type CELL-LINE
Organism Homo sapiens

Publication

Pleiotropic effects of a mitochondrion-targeted glutathione reductase inhibitor on restraining tumor cells.
Zhang R, Xiao N, Xu Q, Gong Q, Kong F, Jiang H.
Eur J Med Chem (2023) 248 : 115069 -115069
PubMed 36610249 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.09 5.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5425052 1 5.09
CHEMBL5403853 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5425052 IC50 = 8200.0 nM 5.09
CHEMBL5403853 IC50 > 50000.0 nM -