Assay Detail
Binding
CHEMBL5327700
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of ATX in human blood
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Tissue | Blood |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent research advances in ATX inhibitors: An overview of primary literature.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.03 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5425421 | — | — | 1 | 8.05 |
| CHEMBL4642052 | — | — | 1 | 8.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5425421 | — | IC50 | = | 8.9 | nM | 8.05 |
| CHEMBL4642052 | — | IC50 | = | 9.7 | nM | 8.01 |