Assay Detail
Binding
CHEMBL5333638
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of telomerase activity in human NCI-H1993 cells by droplet-digital TRAP PCR assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | NCI-H1993 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Telomerase: A prominent oncological target for development of chemotherapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.74 | 6.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL372764 | PERIFOSINE | 3.0 | 1 | 6.74 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL372764 | PERIFOSINE | IC50 | = | 184.0 | nM | 6.74 |