Assay Detail
Binding
CHEMBL5337165
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of KDM2A (unknown origin)
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Focused Screening Identifies Different Sensitivities of Human TET Oxygenases to the Oncometabolite 2-Hydroxyglutarate.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | - | - |
| Ki | 1 | 4.13 | 4.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1614745 | — | — | 2 | 4.13 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1614745 | — | Ki | = | 74000.0 | nM | 4.13 |
| CHEMBL1614745 | — | IC50 | = | 106000.0 | nM | - |