Assay Detail
Binding
CHEMBL5340519
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Binding affinity to G-quadruplex DNA c-kit1 (unknown origin) by fluorescence spectroscopic analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Not specified |
| Confidence | 3 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Development and Characterization of Benzoselenazole Derivatives as Potent and Selective <i>c-MYC</i> Transcription Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 5.11 | 5.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5433462 | — | — | 1 | 5.19 |
| CHEMBL5428440 | — | — | 1 | 5.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5433462 | — | Kd | = | 6500.0 | nM | 5.19 |
| CHEMBL5428440 | — | Kd | = | 9600.0 | nM | 5.02 |