Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5345015

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to CB2 receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cannabinoid receptor 2 (CHEMBL253)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of 4-(1,2,4-Oxadiazol-5-yl)azepan-2-one Derivatives as a New Class of Cannabinoid Type 2 Receptor Agonists for the Treatment of Inflammatory Pain.
Nan J, Liu J, Lin G, Zhang S, Xia A, Zhou P, Zhou Y, Zhang J, Zhao J, Zhang S, Huang C, Wang Y, Hu Q, Chen J, Xiang M, Yang X, Yang S.
J Med Chem (2023) 66 : 3460 -3483
PubMed 36821347 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.47 8.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL408430 1 8.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL408430 Ki = 3.4 nM 8.47