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Assay Detail

CHEMBL5347344

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Coxsackievirus 21 infected in human HeLa cells assessed as reduction of virus induced cytopathic effect incubated for 3 days by MTS assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Coxsackievirus A21
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

Coxsackievirus A21 (CHEMBL613553)
Type ORGANISM
Organism Coxsackievirus A21

Publication

Rational design of novel nucleoside analogues reveals potent antiviral agents for EV71.
Salerno M, Varricchio C, Bevilacqua F, Jochmans D, Neyts J, Brancale A, Ferla S, Bassetto M.
Eur J Med Chem (2023) 246 : 114942 -114942
PubMed 36455356 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 6 4.48 4.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5409037 1 4.70
CHEMBL5434203 1 4.50
CHEMBL389706 1 4.44
CHEMBL5399680 1 4.26
CHEMBL5409662 1 -
CHEMBL5405401 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5409037 EC50 = 19900.0 nM 4.70
CHEMBL5434203 EC50 = 31700.0 nM 4.50
CHEMBL389706 EC50 = 36400.0 nM 4.44
CHEMBL5399680 EC50 = 54600.0 nM 4.26
CHEMBL5409662 EC50 > 100000.0 nM -
CHEMBL5405401 EC50 > 100000.0 nM -