Assay Detail
Binding
CHEMBL5348488
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Inhibition of LTC4 (unknown origin)
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Treatment of allergy: Overview of synthetic anti-allergy small molecules in medicinal chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 6.68 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5417047 | — | — | 1 | 8.70 |
| CHEMBL5432381 | — | — | 1 | 8.30 |
| CHEMBL5400001 | — | — | 1 | 5.80 |
| CHEMBL144830 | — | — | 1 | 5.30 |
| CHEMBL144604 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5417047 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5432381 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL5400001 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL144830 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL144604 | — | IC50 | = | 5000.0 | nM | 5.30 |