Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5357115

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of NDM-1 in Escherichia coli assessed as reduction in imipenem hydrolytic activity
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Escherichia coli
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Beta-lactamase NDM-1 (CHEMBL4295540)
Type SINGLE PROTEIN
Organism Escherichia coli

Publication

Small-molecule inhibitors of bacterial-producing metallo-β-lactamases: insights into their resistance mechanisms and biochemical analyses of their activities.
Ayipo YO, Chong CF, Mordi MN.
RSC Med Chem (2023) 14 : 1012 -1048
PubMed 37360393 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.00 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5396807 1 5.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5396807 IC50 = 10000.0 nM 5.00