Assay Detail
Functional
CHEMBL5358979
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Immunosuppressive activity in mouse splenocyte assessed as reduction in LPS-induced mouse B-cell proliferation
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | Splenocyte |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Diaporaustalides A-L, Austalide Meroterpenoids from a Plant Endophytic <i>Diaporthe</i> sp.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 4.96 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | 4.0 | 1 | 6.00 |
| CHEMBL5439186 | — | — | 1 | 5.42 |
| CHEMBL5422386 | — | — | 1 | 5.17 |
| CHEMBL5411073 | — | — | 1 | 5.07 |
| CHEMBL5422739 | — | — | 1 | 4.77 |
| CHEMBL5405078 | — | — | 1 | 4.51 |
| CHEMBL5423936 | — | — | 1 | 4.41 |
| CHEMBL5416554 | — | — | 1 | 4.36 |
| CHEMBL5432682 | — | — | 1 | - |
| CHEMBL5434311 | — | — | 1 | - |
| CHEMBL5421353 | — | — | 1 | - |
| CHEMBL5413917 | — | — | 1 | - |
| CHEMBL5409295 | — | — | 1 | - |
| CHEMBL160 | CYCLOSPORINE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5439186 | — | IC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL5422386 | — | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL5411073 | — | IC50 | = | 8500.0 | nM | 5.07 |
| CHEMBL5422739 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL5405078 | — | IC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL5423936 | — | IC50 | = | 39000.0 | nM | 4.41 |
| CHEMBL5416554 | — | IC50 | = | 44000.0 | nM | 4.36 |
| CHEMBL5432682 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5434311 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5421353 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5413917 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5409295 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL160 | CYCLOSPORINE | IC50 | - | — | - |