Assay Detail
Binding
CHEMBL5359055
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]CP55940 from human CB2 receptor expressed in Sf9 cell membranes assessed as inhibition constant incubated for 90 mins by by scintillation counter analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Sf9 |
| Subcellular | Membrane |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
A Simple Chiral <sup>1</sup>H NMR Method for the Discrimination of (<i>R</i>)- and (<i>S</i>)-Cannabichromene in Complex Natural Mixtures and Their Effects on TRPA1 Activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.58 | 6.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL422704 | CANNABICHROMENE | — | 1 | 6.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL422704 | CANNABICHROMENE | Ki | = | 260.0 | nM | 6.58 |