Assay Detail
Binding
CHEMBL5360494
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Binding affinity to CB2 receptor (unknown origin) assessed as inhibition constant
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and Evaluation of Natural and Unnatural Tetrahydrocannabiorcol for Its Potential Use in Neuropathologies.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.32 | 7.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL465 | DRONABINOL | 4.0 | 1 | 7.44 |
| CHEMBL2387541 | TETRAHYDROCANNABIVARIN | 2.0 | 1 | 7.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL465 | DRONABINOL | Ki | = | 36.4 | nM | 7.44 |
| CHEMBL2387541 | TETRAHYDROCANNABIVARIN | Ki | = | 62.8 | nM | 7.20 |