Assay Detail
Binding
CHEMBL5371701
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human NSD3 SET domain assessed as reduction in H3K36 methylation
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Histone-lysine N-methyltransferase NSD3 (CHEMBL3108646) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
NSD3: Advances in cancer therapeutic potential and inhibitors research.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.02 | 4.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1895209 | — | — | 1 | 4.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1895209 | — | IC50 | = | 95000.0 | nM | 4.02 |