Assay Detail
Binding
CHEMBL5372963
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Binding affinity to human Y4R under sodium free condition
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 9.10 | 9.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5411178 | — | — | 1 | 9.17 |
| CHEMBL5428989 | — | — | 1 | 9.17 |
| CHEMBL5407336 | — | — | 1 | 8.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5411178 | — | Kd | = | 0.67 | nM | 9.17 |
| CHEMBL5428989 | — | Kd | = | 0.67 | nM | 9.17 |
| CHEMBL5407336 | — | Kd | = | 1.1 | nM | 8.96 |