Assay Detail
Binding
CHEMBL5378339
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Inhibition of His6-tagged KIND2 (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence polarization method
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of Inhibitory Fragments That Selectively Target Spire2-FMN2 Interaction.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 26 | 3.55 | 4.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5394576 | — | — | 1 | 4.21 |
| CHEMBL2393341 | — | — | 1 | 3.99 |
| CHEMBL99254 | — | — | 1 | 3.57 |
| CHEMBL236491 | — | — | 1 | 3.44 |
| CHEMBL316953 | — | — | 1 | 3.35 |
| CHEMBL235241 | — | — | 1 | 3.25 |
| CHEMBL581588 | — | — | 1 | 3.03 |
| CHEMBL460418 | — | — | 1 | - |
| CHEMBL44789 | — | — | 1 | - |
| CHEMBL1241726 | — | — | 1 | - |
| CHEMBL236696 | — | — | 1 | - |
| CHEMBL31000 | — | — | 1 | - |
| CHEMBL98114 | — | — | 1 | - |
| CHEMBL5414257 | — | — | 1 | - |
| CHEMBL5426817 | — | — | 1 | - |
| CHEMBL5414970 | — | — | 1 | - |
| CHEMBL5414019 | — | — | 1 | - |
| CHEMBL5403742 | — | — | 1 | - |
| CHEMBL5414961 | — | — | 1 | - |
| CHEMBL2393338 | — | — | 1 | - |
| CHEMBL2393337 | — | — | 1 | - |
| CHEMBL5399645 | — | — | 1 | - |
| CHEMBL5403660 | — | — | 1 | - |
| CHEMBL5402421 | — | — | 1 | - |
| CHEMBL5430068 | — | — | 1 | - |
| CHEMBL5407372 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5394576 | — | IC50 | = | 62000.0 | nM | 4.21 |
| CHEMBL2393341 | — | IC50 | = | 103000.0 | nM | 3.99 |
| CHEMBL99254 | — | IC50 | = | 268000.0 | nM | 3.57 |
| CHEMBL236491 | — | IC50 | = | 362000.0 | nM | 3.44 |
| CHEMBL316953 | — | IC50 | = | 448000.0 | nM | 3.35 |
| CHEMBL235241 | — | IC50 | = | 565000.0 | nM | 3.25 |
| CHEMBL581588 | — | IC50 | = | 938000.0 | nM | 3.03 |
| CHEMBL460418 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL44789 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL1241726 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL236696 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL31000 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL98114 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5414257 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5426817 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5414970 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5414019 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5403742 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5414961 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL2393338 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL2393337 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5399645 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5403660 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5402421 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5430068 | — | IC50 | > | 2500000.0 | nM | - |
| CHEMBL5407372 | — | IC50 | > | 2500000.0 | nM | - |