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Assay Detail

CHEMBL5379112

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Antiproliferative activity against mouse NIH3T3 cells assessed as inhibition of cell growth measured after 48 hrs by MTT assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Mus musculus
Cell Type NIH3T3
Confidence 1 — Organism
Curated By Autocuration

Target

NIH3T3 (CHEMBL614822)
Type CELL-LINE
Organism Mus musculus

Publication

Pioneering 4,11-Dioxo-4,11-dihydro-1<i>H</i>-anthra[2,3-<i>d</i>]imidazol-3-ium Compounds as Promising Survivin Inhibitors by Targeting ILF3/NF110 for Cancer Therapy.
Yuan J, Liu Z, Dong Y, Gao F, Xia X, Wang P, Luo Y, Zhang Z, Yan D, Zhang W.
J Med Chem (2023) 66 : 16843 -16868
PubMed 38079530 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.86 4.87

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2105734 SEPANTRONIUM BROMIDE 2.0 1 4.87
CHEMBL5437193 1 4.85
CHEMBL5411686 1 4.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2105734 SEPANTRONIUM BROMIDE IC50 = 13600.0 nM 4.87
CHEMBL5437193 IC50 = 14200.0 nM 4.85
CHEMBL5411686 IC50 = 14000.0 nM 4.85