Assay Detail
Binding
CHEMBL5381304
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to BRD4 bromodomain 1 (unknown origin) assessed as dissociation constant
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent Advances on Small-Molecule Bromodomain-Containing Histone Acetyltransferase Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.00 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3752296 | — | — | 1 | 6.00 |
| CHEMBL5394573 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3752296 | — | Kd | = | 1010.0 | nM | 6.00 |
| CHEMBL5394573 | — | Kd | > | 40000.0 | nM | - |