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Assay Detail

CHEMBL5382181

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of PIM2 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Serine/threonine-protein kinase pim-2 (CHEMBL4523)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Strategies of Targeting CK2 in Drug Discovery: Challenges, Opportunities, and Emerging Prospects.
Chen Y, Wang Y, Wang J, Zhou Z, Cao S, Zhang J.
J Med Chem (2023) 66 : 2257 -2281
PubMed 36745746 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.47 6.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL270722 1 6.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL270722 IC50 = 340.0 nM 6.47