Assay Detail
Binding
CHEMBL5390058
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PD-L1 (unknown origin) by HTRF assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Progress in small-molecule inhibitors targeting PD-L1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 9.50 | 9.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5413429 | — | — | 1 | 9.68 |
| CHEMBL5398154 | — | — | 1 | 9.32 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5413429 | — | IC50 | = | 0.21 | nM | 9.68 |
| CHEMBL5398154 | — | IC50 | = | 0.48 | nM | 9.32 |