Assay Detail
Binding
CHEMBL5446169
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Affinity Biochemical interaction: (Biochemical assay (LPA measurement)) EUB0001066a ENPP2
1
Total Activities
1
Compounds Tested
1
Activity Types
3
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | Affinity biochemical assay |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Affinity Biochemical Literature for EUbOPEN Chemogenomic Library
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.05 | 5.05 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Mode of action | Mode of action | - | — | Negative control for BI-2545 |
| Protein family | Protein family | - | — | PDE |
| Recommended concentration | Recommended concentration | 1.0 | uM | — |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4552354 | BI 3017 | — | 1 | 5.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4552354 | BI 3017 | IC50 | = | 8900.0 | nM | 5.05 |