Assay Detail
Binding
CHEMBL5481235
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Selectivity interaction (Biochemical dose-response assay (Carna Biosciences)) EUB0001326b CDK9
1
Total Activities
1
Compounds Tested
1
Activity Types
1
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | Selectivity assay |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Selectivity Literature for EUbOPEN Chemogenomic Library
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 9.00 | 9.00 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Protein family | Protein family | - | — | Protein kinase |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1.0 | nM | 9.00 |