Assay Detail
Binding
CHEMBL5505737
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of IRAP (unknown origin) using L-pNA as substrate
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Interleukin-1 receptor antagonist protein (CHEMBL4523191) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
ERAP Inhibitors in Autoimmunity and Immuno-Oncology: Medicinal Chemistry Insights.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.68 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL83148 | PHENYL(PHENYLSULFONYL)AMINE | — | 1 | 5.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL83148 | PHENYL(PHENYLSULFONYL)AMINE | IC50 | = | 2100.0 | nM | 5.68 |