Assay Detail
Binding
CHEMBL5514067
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of ABL (unknown origin) incubated for 1 hr by ADP-Glo assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Research progress of DDR1 inhibitors in the treatment of multiple human diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.24 | 8.03 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4175086 | — | — | 1 | 8.03 |
| CHEMBL2336015 | — | — | 1 | 6.45 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4175086 | — | IC50 | = | 9.4 | nM | 8.03 |
| CHEMBL2336015 | — | IC50 | = | 355.0 | nM | 6.45 |